Identification of novel protein kinase CK1 delta (CK1δ) inhibitors through structure-based virtual screening
Articolo
Data di Pubblicazione:
2008
Tipologia CRIS:
1.1 Articolo in rivista
Keywords:
Kinase inhibitors; Molecular docking; Protein kinase CK1 delta; Structure-based virtual screening; Anthraquinones; Casein Kinase I; Chemistry, Pharmaceutical; Computer Simulation; Drug Design; Drug Evaluation, Preclinical; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Molecular Conformation; Phosphorylation; Protein Isoforms; Software; Tyrosine; 3003; Drug Discovery3003 Pharmaceutical Science; Organic Chemistry; Molecular Medicine; Molecular Biology; Clinical Biochemistry; Biochemistry
Elenco autori:
Cozza, Giorgio; Gianoncelli, Alessandra; Montopoli, Monica; Caparrotta, Laura; Venerando, Andrea; Meggio, Flavio; Pinna, Lorenzo A.; Zagotto, Giuseppe; Moro, Stefano
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